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Plasma pharmacokinetic parameters
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Image Search Results


Plasma pharmacokinetic parameters

Journal: Clinical and Translational Science

Article Title: A thorough QTc study to evaluate the effects of oral rilzabrutinib administered alone and with ritonavir in healthy subjects

doi: 10.1111/cts.13271

Figure Lengend Snippet: Plasma pharmacokinetic parameters

Article Snippet: Plasma concentrations of rilzabrutinib and moxifloxacin were quantified by Alturas Analytics Inc. (Moscow, ID, USA).

Techniques: Clinical Proteomics, Positive Control

Effects of rilzabrutinib on electrocardiogram (ECG) parameters across timepoints over 24 h after administration of rilzabrutinib 400 mg (blue line), rilzabrutinib 400 mg + ritonavir 100 mg (red line), placebo (gray line), or moxifloxacin (green line) in Part B. (a) Change from baseline in heart rate (ΔHR) and (b) mean change from baseline in QTcF interval over time using Fridericia's formula (ΔQTcF)

Journal: Clinical and Translational Science

Article Title: A thorough QTc study to evaluate the effects of oral rilzabrutinib administered alone and with ritonavir in healthy subjects

doi: 10.1111/cts.13271

Figure Lengend Snippet: Effects of rilzabrutinib on electrocardiogram (ECG) parameters across timepoints over 24 h after administration of rilzabrutinib 400 mg (blue line), rilzabrutinib 400 mg + ritonavir 100 mg (red line), placebo (gray line), or moxifloxacin (green line) in Part B. (a) Change from baseline in heart rate (ΔHR) and (b) mean change from baseline in QTcF interval over time using Fridericia's formula (ΔQTcF)

Article Snippet: Plasma concentrations of rilzabrutinib and moxifloxacin were quantified by Alturas Analytics Inc. (Moscow, ID, USA).

Techniques:

Placebo‐corrected change from baseline QTcF (ΔΔQTcF) <xref ref-type= a (Part B)" width="100%" height="100%">

Journal: Clinical and Translational Science

Article Title: A thorough QTc study to evaluate the effects of oral rilzabrutinib administered alone and with ritonavir in healthy subjects

doi: 10.1111/cts.13271

Figure Lengend Snippet: Placebo‐corrected change from baseline QTcF (ΔΔQTcF) a (Part B)

Article Snippet: Plasma concentrations of rilzabrutinib and moxifloxacin were quantified by Alturas Analytics Inc. (Moscow, ID, USA).

Techniques:

Treatment‐related treatment‐emergent adverse events (Part B)

Journal: Clinical and Translational Science

Article Title: A thorough QTc study to evaluate the effects of oral rilzabrutinib administered alone and with ritonavir in healthy subjects

doi: 10.1111/cts.13271

Figure Lengend Snippet: Treatment‐related treatment‐emergent adverse events (Part B)

Article Snippet: Plasma concentrations of rilzabrutinib and moxifloxacin were quantified by Alturas Analytics Inc. (Moscow, ID, USA).

Techniques: Infection